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   CAS NO.    Products Name
   1009298-59-2 AZD2014  more...
   AZD2014 is a close analogue of AZD8055 and a selective inhibitor of mTOR kinase. AZD2014 has greater inhibitory activity against mTORC1 compared to rapamycin: AZD2014 decreases p4EBP1 T...
   1009298-09-2 AZD8055  more...
   Biological Activity of AZD8055: AZD8055 is a potent, selective, and orally bioavailable ATP-competitive mTOR kinase inhibitor with an IC50 of 0.8 nM. It inhibits the phosphorylation of...
   572924-54-0 Deforolimus  more...
   Deforolimus (Ridaforolimus) is a small-molecule inhibitor of mTOR. It is an immunosuppressant for the treatment of certain cancers. Blocking mTOR creates a starvation-like effect in can...
   159351-69-6 Everolimus  more...
   Everolimus(RAD001), is a 40-O-(2-hydroxyethyl) derivative of rapamycin with immunosuppressant and anti-angiogenic properties, which exhibits improved aqueous solubility relative to the ...
   1224844-38-5 INK 128 (MLN0128)  more...
   INK 128 exhibits an enzymatic inhibition activity against mTOR and more than 100-fold selectivity to PI3K kinases. As TORC1/2 inhibitor, INK 128 inhibits both the phosphorylation of S6 ...
   938440-64-3 ku0063794  more...
   Ku-0063794 is a specific inhibitor of mTOR, which inhibits both mTORC1 and mTORC2 with an IC50 of approximately 10 nM, but does not suppress the activity of 76 other protein kinases or ...
   1092351-67-1 PP242  more...
   PP242 is a novel potent and selective mTOR inhibitor with an IC50 of 8 nM. PP242 also shows residual (micromolar) activity against panel of tyrosine kinases. But PP242 was much less act...
   53123-88-9 Rapamycin  more...
   rapamycin inhibited the proliferation of primary bone marrow cells induced by IL-3, GM-CSF, KL, or a complex mixture of factors present in cell-conditioned media. Rapamycin also inhibit...
   162635-04-3 Temsirolimus  more...
   Temsirolimus (also known as CCI-779) is a recently developed mTOR inhibitor, with improved aqueous solubility and more favorable pharmaceutical properties compared with the parent compo...
   1144068-46-1 WYE 125132  more...
   WYE-125132 is a highly potent, ATP-competitive and specific mTOR kinase inhibitor with an IC50 of 0.19 nM. WYE-125132 blocked the activity of the both of mTORC1 and mTORC2 in various mo...

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