AP-III-a4 ENOblock

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Chemical Information

Product name：AP-III-a4 ENOblock	Purity：98% min
CAS NO：1177827-73-4	Solubility：
Molecular Formula：C₃₁H₄₃FN₈O₃	Package：Package according to customer requirements
Molecular Weight：594.723	Storage：Store at -20℃

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Remarks

ENOblock(AP-III-a4) is a novel small molecule which is the first, nonsubstrate analogue that directly binds to enolase and inhibits its activity (IC50=0.576 uM); inhibit cancer cell metastasis in vivo.

References

[1]. Da-Woon Jung, et al. A Unique Small Molecule Inhibitor of Enolase Clarifies Its Role in Fundamental Biological Processes.ACS Chem. Biol., 2013, 8 (6), pp 1271–1282