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Ro 25-6981 Maleate

Ro 25-6981 Maleate  1312991-76-6
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Chemical Information
Product name:Ro 25-6981 Maleate Purity:98% min
CAS NO:1312991-76-6 Solubility:DMSO : ≥ 61 mg/mL (133.91 mM)
Molecular Formula:C26H33NO6 Package:Package according to customer requirements
Molecular Weight:455.543 Storage:Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Quality control
Ro 25-6981 maleate is a highly potent and selective blocker of N-methyl-D-aspartate receptors containing the NR2B subunit. Ro 25-6981 inhibited 3H-MK-801 binding to rat forebrain membranes in a biphasic manner with IC50 values of 0.003 microM and 149 microM for high- (about 60%) and low-affinity sites, respectively. NMDA receptor subtypes expressed in Xenopus oocytes were blocked with IC50 values of 0.009 microM and 52 microM for the subunit combinations NR1C & NR2B and NR1C & NR2A, respectively, which indicated a >5000-fold selectivity.
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