ARN272

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Chemical Information

Product name：ARN272	Purity：98% min
CAS NO：488793-85-7	Solubility：
Molecular Formula：C₂₇H₂₀N₄O₂	Package：Package according to customer requirements
Molecular Weight：432.473	Storage：-20 ℃

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Remarks

ARN272 is a FAAH-like anandamide transporter (FLAT) inhibitor. ARN272 attenuates nausea-induced behaviour in rats, and vomiting in shrews (Suncus murinus). The anandamide transport inhibition by ARN272 tonically activates CB1 receptors and as such produces a type of indirect agonism to regulate toxin-induced nausea and vomiting.

References

[1]. O'Brien LD, et al. Anandamide transport inhibition by ARN272 attenuates nausea-induced behaviour in rats, and vomiting in shrews (Suncus murinus). Br J Pharmacol. 2013 Nov;170(5):1130-6.