CID 2011756

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Chemical Information

Product name：CID 2011756	Purity：98% min
CAS NO：638156-11-3	Solubility：DMSO : 20 mg/mL (50.39 mM)
Molecular Formula：C₂₂H₂₁ClN₂O₃	Package：Package according to customer requirements
Molecular Weight：396.867	Storage：Store at -20℃

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Remarks

CID 2011756 is an ATP competitive PKD inhibitor, with an IC50 of 3.2 µM for PKD1 in cell free assay, and also shows cellular pan-PKD inhibitory activity against PKD2 and PKD3 (IC50, 0.6 and 0.7 µM, respectively). CID 2011756 also has antitumor activity.

References

[1]. Sharlow ER, et al. Discovery of diverse small molecule chemotypes with cell-based PKD1 inhibitory activity. PLoS One. 2011;6(10):e25134.