Acetorphan Racecadotril

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Chemical Information

Product name：Acetorphan Racecadotril	Purity：98% min
CAS NO：81110-73-8	Solubility：DMSO : ≥ 100 mg/mL (259.42 mM)
Molecular Formula：C₂₁H₂₃NO₄S	Package：Package according to customer requirements
Molecular Weight：385.48	Storage：Store at -20℃

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Remarks

Racecadotril, also known as acetorphan, is an antidiarrheal drug which acts as a peripherally acting enkephalinase inhibitor. Unlike other opioid medications used to treat diarrhea, which reduce intestinal motility, racecadotril has an antisecretory effect-it reduces the secretion of water and electrolytes into the intestine.

Properties:
Appearance & Physical State: White to off-white crystalline power
Density: 1.206
Melting Point: 89ºC
Boiling Point: 574.5ºC at 760 mmHg
Flash Point: 301.2ºC
Refractive Index: 1.601

Opioid Receptor Inhibitors Related Products:

JTC-801; Naltrexone HCl; Alvimopan; Trimebutine Maleate Salt; Trimebutine

References

[1]. Marion Eberlin, Tobias Mück, Martin C. Michel, et al. A Comprehensive Review of the Pharmacodynamics, Pharmacokinetics, and Clinical Effects of the Neutral Endopeptidase Inhibitor Racecadotril. Front Pharmacol. 2012; 3: 93.

[2]. Wu HT, Chang CK, Cheng KC, et al. Increase of plasma insulin by racecadotril, an inhibitor of enkephalinase, in Wistar rats. Horm Metab Res. 2010 Apr;42(4):261-7.