Teneligliptin hydrobromide

Size	Price	Stock	Quantity
Get Quotation Now Add to Cart Bulk Inquiry

Shipping and handling fee USD40, Free delivery is qualified when the total value of your order exceeds USD500.If the item is temporarily out of stock. Please email to order@pharm-intermediates.com,we will inform you when we have it in stock.

Chemical Information

Product name：Teneligliptin hydrobromide	Purity：98% min
CAS NO：906093-29-6	Solubility：DMSO : ≥ 100 mg/mL (159.02 mM); H2O : ≥ 200 mg/mL (318.04 mM)
Molecular Formula：C₄₄H₆₅Br₅N₁₂O₂S₂	Package：Package according to customer requirements
Molecular Weight：1257.720	Storage：Store at -20℃

Quality control

COA

Remarks

Teneligliptin (MP-513) hydrobromide is a potent chemotype prolylthiazolidine-based DPP-4 inhibitor, which competitively inhibits human plasma, rat plasma, and human recombinant DPP-4 in vitro, with IC50s of approximately 1 nM.

DPP-4 Inhibitor Related Products:

Alogliptin benzoate; Sitagliptin phosphate monohydrate; Linagliptin; Vildagliptin; Saxagliptin; Trelagliptin succinate; Omarigliptin; Saxagliptin hydrate; Trelagliptin; Saxagliptin HCL ; Alogliptin

References

[1]. Fukuda-Tsuru S, et al. A novel, potent, and long-lasting dipeptidyl peptidase-4 inhibitor, teneligliptin, improves postprandial hyperglycemia and dyslipidemia after single and repeated administrations. Eur J Pharmacol. 2012 Dec 5;696(1-3):194-202.

[2]. Ideta T, et al. The Dipeptidyl Peptidase-4 Inhibitor Teneligliptin Attenuates Hepatic Lipogenesis via AMPK Activation in Non-Alcoholic Fatty Liver Disease Model Mice. Int J Mol Sci. 2015 Dec 8;16(12):29207-18.