Product :
MPC-3100
Shipping and handling fee USD40, Free delivery is qualified when the total value of your order exceeds USD500.If the item is temporarily out of stock. Please email to order@pharm-intermediates.com,we will inform you when we have it in stock.
Chemical Information
Product name:MPC-3100 |
Purity:98% min |
CAS NO:958025-66-6 |
Solubility:Soluble in DMSO |
Molecular Formula:C22H25BrN6O4S |
Package:Package according to customer requirements |
Molecular Weight:549.441 |
Storage:Store at -20℃ |
Remarks
MPC-3100 is a n orally bioavailable, synthetic, second-generation small-molecule inhibitor of heat shock protein 90 (Hsp90) with potential antineoplastic activity. Hsp90 inhibitor MPC-3100 selectively binds to Hsp90, thereby inhibiting its chaperone function and promoting the degradation of oncogenic signaling proteins involved in tumor cell proliferation and survival; this agent may inhibit the growth and survival of a wide variety of cancer cell types.
References
1: Sidera K, Patsavoudi E. HSP90 inhibitors: current development and potential in cancer therapy. Recent Pat Anticancer Drug Discov. 2014 Jan;9(1):1-20. Review. PubMed PMID: 23312026.