JMS-17-2 is a potent and selective CX3CR1 antagonist with an IC50 of 0.32 nM.
Chemical Name:
5-(3-(4-(4-chlorophenyl)piperidin-1-yl)propyl)pyrrolo[1,2-a]quinoxalin-4(5H)-one
GPR Inhibitors Related Prodcuts:
Timapiprant; GSK137647A; CID 1375606; APD668