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Product :

CPI-637

CPI-637 1884712-47-3
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Chemical Information
Product name:CPI-637 Purity:98% min
CAS NO:1884712-47-3 Solubility:DMSO : 12.5 mg/mL (32.35 mM)
Molecular Formula:C22H22N6O Package:Package according to customer requirements
Molecular Weight:386.450 Storage:Store at -20℃
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Remarks

CPI-637 is a potent and selective CBP/ EP300 bromodomain inhibitor. The biochemical potency of CPI-637 translated well into cells (CBP BRET EC50 = 0.3 μM). CPI-637 demonstrated a >700-fold selectivity over the BET family of bromodomains (BRD4 IC50 = 11.0 ± 0.6 μM). CPI-637 inhibits MYC expression in AMO-1 cells (EC50 = 0.60 μM). CBP and EP300 are highly homologous, bromodomain-containing transcription coactivators involved in numerous cellular pathways relevant to oncology.

 

 

 

Histone Acetyltransferase Inhibitors Related Prodcuts:

C646; Curcumin; ReModelin Hydrobromide; ReModelin; WM-1119

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.
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