MM-102

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Chemical Information

Product name：MM-102	Purity：99% min
CAS NO：1417329-24-8	Solubility：Soluble in DMSO
Molecular Formula：C₃₅H₄₉F₂N₇O₄	Package：Package according to customer requirements
Molecular Weight：669.805	Storage：Store at -20℃

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Remarks

MM-102 is a potent WDR5/MLL interaction inhibitor, achieves IC50 = 2.4 nM with an estimated Ki < 1 nM in WDR5 binding assay, which is >200 times more potent than the ARA peptide.

Histone Methyltransferase Inhibitors Related Products:

EPZ005687; GSK343; Tazemetostat; UNC1999; SGC0946; SGC2085; OICR-9429; HLCL-61 HCL; GSK591; SGC707; GSK503; EPZ015666; PFI-2 HCl; UNC0642; UNC0638; GSK-126; EPZ004777; GSK3326595; LLY-507; BRD4770 ; Pinometostat

References

[1]. Karatas H, et al. High-affinity, small-molecule peptidomimetic inhibitors of MLL1/WDR5 protein-protein interaction. J Am Chem Soc. 2013, 135(2), 669-682.