Y-25130 Azasetron hydrochloride

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Chemical Information

Product name：Y-25130 Azasetron hydrochloride	Purity：99% min
CAS NO：123040-16-4	Solubility：H2O : ≥ 3.9 mg/mL (10.10 mM)
Molecular Formula：C₁₇H₂₁Cl₂N₃O₃	Package：Package according to customer requirements
Molecular Weight：386.273	Storage：Store at -20℃

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Remarks

Azasetron HCl is a selective 5-HT3 receptor antagonist with IC50 of 0.33 nM used in the management of nausea and vomiting induced by cancer chemotherapy.

Properties:

Boiling Point 558ºC at 760 mmHg
Flash Point 291.2ºC

5-HT Receptor Inhibitors Related Products:

RS-127445; Asenapine Maleate; WAY-100635 Maleate; WAY-100635 maleate salt; Vortioxetine; Vortioxetine hydrobromide; Blonanserin; Intepirdine; Sertraline HCl; Lamotrigine; Iloperidone

References

[1]. Sato, N., et al., Antagonistic activity of Y-25130 on 5-HT3 receptors. Jpn J Pharmacol, 1992. 59(4): p. 443-8.

[2]. Haga, K., et al., The effects of orally administered Y-25130, a selective serotonin3-receptor antagonist, on chemotherapeutic agent-induced emesis. Jpn J Pharmacol, 1993. 63(3): p. 377-83.