CGS-15943

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Chemical Information

Product name：CGS-15943	Purity：98% min
CAS NO：104615-18-1	Solubility：DMSO : 12.22 mg/mL (42.77 mM)
Molecular Formula：C₁₃H₈ClN₅O	Package：Package according to customer requirements
Molecular Weight：285.689	Storage：-20℃

Quality control

Remarks

CGS15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor with Ki of 3.5 nM, 4.2 nM, 16 nM, and 50 nM for human A1, A2A, A2B, and A3 Adenosine Receptors in transfected CHO cells, respectively.

Properties:

Appearance & Physical State: solid

Density: 1.72 g/cm3

Boiling Point: 566.6ºC at 760 mmHg

Flash Point: 296.5ºC

Refractive Index: 1.84

Vapor Pressure: 7.4E-13mmHg at 25°C

Adenosine Receptor Related Products:

ZM241385; Preladenant; Reversine; SCH-58261; Istradefylline; Regadenoson; Tozadenant; Adenosine amine congener (ADAC); CGS-21680; CGS-21680 HCl; Vipadenant

References

[1]. Gao Y, et al. CGS 15943, an adenosine A2 receptor antagonist, reduces cerebral ischemic injury in the Mongolian gerbil. Life Sci. 1994;55(3):PL61-5.

[2]. Klotz KN, et al. Adenosine receptors and their ligands. Naunyn Schmiedebergs Arch Pharmacol. 2000 Nov;362(4-5):382-91.