TD-4208 Revefenacin

Size	Price	Stock	Quantity
Get Quotation Now Add to Cart Bulk Inquiry

Shipping and handling fee USD40, Free delivery is qualified when the total value of your order exceeds USD500.If the item is temporarily out of stock. Please email to order@pharm-intermediates.com,we will inform you when we have it in stock.

Chemical Information

Product name：TD-4208 Revefenacin	Purity：98% min
CAS NO：864750-70-9	Solubility：DMSO : ≥ 125 mg/mL (209.12 mM)
Molecular Formula：C₃₅H₄₃N₅O₄	Package：Package according to customer requirements
Molecular Weight：597.747	Storage：Store at -20℃

Quality control

Remarks

Revefenacin, also known as TD-4208; GSK-1160724, is a long-acting muscarinic receptor antagonist and may be potentially useful for the treatment of respiratory disease.

Chemical Name:

biphenyl-2-ylcarbamic acid 1-(2-{[4-(4-carbamoylpiperidin-1-ylmethyl)benzoyl]methylamino}ethyl)piperidin-4-ylester

AChR Inhibitors Related Products:

Donepezil Hcl; (-)-Huperzine A; PNU-120596; Scopolamine hydrobromide; Rivastigmine Tartrate; Darifenacin hydrobromide; Vinblastine sulfate; Tolterodine tartrate; Amfebutamone hydrochloride; Solifenacin; Solifenacin succinate; Trospium chloride; Pyridostigmine bromide; Varenicline; Imidafenacin

References

[1]. Steinfeld T, et al. In vitro characterization of TD-4208, a lung-selective and long-acting muscarinic antagonist bronchodilator (Abstract). Am J Respir Crit Care Med 179:A4553.

[2]. Pulido-Rios MT, et al. In vivo pharmacological characterization of TD-4208, a novel lung-selective inhaled muscarinic antagonist with sustained bronchoprotective effect in experimental animal models. J Pharmacol Exp Ther. 2013 Aug;346(2):241-50.