MRS1845 is a selective store-operated calcium (SOC) channel inhibitor with an IC50 of 1.7 μM. MRS1845 is an ORAI1 inhibitor.
Chemical Name:
5-O-ethyl 3-O-methyl 2,6-dimethyl-4-(3-nitrophenyl)-1-prop-2-ynyl-4H-pyridine-3,5-dicarboxylate
Properties:
Density: 1.318g/cm3
Boiling Point: 530.8ºC at 760 mmHg
Flash Point: 274.8ºC
Refractive Index: 1.595
Calcium Channel Related Products:
Manidipine 2HCl; Felodipine; Nisoldipine; Fasudil HCl; Cilnidipine; Dronedarone HCl; Clevidipine Butyrate; Efonidipine; Amlodipine; ISX-9 (Isoxazole 9); Gabapentin; Fantofarone; Suvecaltamide (MK-8998); Ziconotide; Catharanthine Tartrate; Bepridil hydrochloride