Trilaciclib is a CDK4/6 inhibitor with IC50s of 1 nM and 4 nM for CDK4 and CDK6, respectively.
Synonyms:
2'-((5-(4-methylpiperazin-1-yl)pyridin-2-yl)amino)-7',8'-dihydro-6'H-spiro(cyclohexane-1,9'-pyrazino(1',2':1,5)pyrrolo(2,3-d)pyrimidin)-6'-one;
G1T28;
Properties:
density: 1.46±0.1 g/cm3(Predicted)
pka: 13.33±0.20(Predicted)
CDK Inhibitors Related Products:
Palbociclib HCl; SNS-032; PF-00562271 Besylate; A-674563; NU6027; 1-NM-PP1; YKL-5-124; OTS964 HCl; Indisulam; Apcin; Palbociclib