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Product :

G007-LK

G007-LK 1380672-07-0
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Chemical Information
Product name:G007-LK Purity:98% min
CAS NO:1380672-07-0 Solubility:DMSO : ≥ 30 mg/mL (56.61 mM)
Molecular Formula:C25H16ClN7O3S Package:Package according to customer requirements
Molecular Weight:529.958 Storage:Store at -20℃
Quality control
COA
Remarks

G007-LK is a potent, "rule of 5" compliant and a metabolically stable TNKS1/2 inhibitor. G007-LK displayed high selectivity toward tankyrases 1 and 2 with biochemical IC50 values of 46 nM and 25 nM, respectively, and a cellular IC50 value of 50 nM combined with an excellent pharmacokinetic profile in mice. G007-LK was first discovered by Dr. Stefan Krauss's team.

 

 

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Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.
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